CCG258208 (hydrochloride)
Catalogue number:
HY-109562A-100mg
Supplier:
Size:
100 mg
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
Purity:
98.05
Molecular Formula:
C24H26ClFN4O4
Molecular Weight:
488.94
Mass Spectrometry:
Reference Materials
Alternative Names:
GRK2-IN-1 (hydrochloride)
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
CCG258208 (GRK2-IN-1) hydrochloride is a potent and selective GRK2 (G protein-coupled receptor kinase 2) inhibitor (IC50=30 nM) while maintaining 230-fold selectivity over GRK5 (IC50=7.09 µM) and more than 2500-fold selectivity over GRK1 (IC50=87.3 µM), PKA, and ROCK1. CCG258208 hydrochloride can be used in heart failure research[1].
