Sograzepide
Catalogue number:
HY-14850-50mg
Supplier:
Size:
50 mg
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
155488-25-8
Purity:
98.28
Molecular Formula:
C28H30N6O3
Molecular Weight:
498.58
Mass Spectrometry:
Reference Materials
Alternative Names:
Netazepide; YF 476; YM-220
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Sograzepide (Netazepide; YF 476; YM-220) is an extremely potent, highly selective and orally active Gastrin/CCK-B antagonist with an IC50 value of 0.1 nM, has inhibitory effect on Gastrin/CCK-A activity with an IC50 of 502 nM[1]. Sograzepide (Netazepide; YF 476; YM-220) replaces the specific binding of [125I]CCK-8 to the rat brain, cloned canine and cloned human Gastrin/CCK-B receptors, with Ki values of 0.068, 0.62 and 0.19 nM, respectively[2].
