Umbralisib (hydrochloride)
Catalogue number:
HY-12279C-50mg
Supplier:
Size:
50 mg
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1532533-78-0
Purity:
99.04
Molecular Formula:
C31H25ClF3N5O3
Molecular Weight:
608.01
Mass Spectrometry:
Reference Materials
Alternative Names:
TGR-1202 hydrochloride; RP5264 hydrochloride
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Umbralisib (TGR-1202) hydrochloride is an orally active, potent and selective dual PI3Kδ and casein kinase-1-ε (CK1ε) inhibitor, with EC50 of 22.2 nM and 6.0 µM, respectively. Umbralisib hydrochloride exhibits unique immunomodulatory effects on chronic lymphocytic leukemia (CLL) T cells. Umbralisib hydrochloride can be used for haematological malignancies reseach[1][2][3][4].
