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Methiothepin (mesylate)

Catalogue number:
HY-107836-1ml
Supplier:
Size:
1 ml
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

74611-28-2

Purity:

99.60

Molecular Formula:

C21H28N2O3S3

Molecular Weight:

452.65

Mass Spectrometry:

Reference Materials

Alternative Names:

Metitepine (mesylate); Ro 8-6837 (mesylate)

Product Description:

Methiothepin (Metitepine) mesylate is a potent and non-selective 5-HT2 receptor antagonist, with pKds of 7.10 (5-HT1A), 7.28 (5HT1B), 7.56 (5HT1C), 6.99 (5HT1D), 7.0 (5-HT5A), 7.8 (5-HT5B), 8.74 (5-HT6), and 8.99 (5-HT7), and pKis of 8.50 (5HT2A), 8.68 (5HT2B), and 8.35 (5HT2C). 10mM