RSM-932A
Catalogue number:
HY-101144-100mg
Supplier:
Size:
100 mg
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
850807-63-5
Purity:
98.44
Molecular Formula:
C46H38Br2Cl2N4
Molecular Weight:
877.53
Mass Spectrometry:
Reference Materials
Alternative Names:
TCD-717
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
RSM-932A (TCD-717) is a specific ChoKα inhibitor with IC50s of 1 and 33 µM for human recombinant ChoKα and ChoKβ enzymes, respectively. RSM-932A acts as the “first in humans” compound targeting ChoKα. RSM-932A is potent in vitro anti-proliferative and in vivo anti-tumoral activity against human xenografts in mice, showing high efficacy with low toxicity profiles[1][2][3].