Zefamenib
Catalogue number:
HY-153714-25mg
Supplier:
Size:
25 mg
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
2938995-50-5
Purity:
98.60
Molecular Formula:
C31H35FN8O2
Molecular Weight:
570.66
Mass Spectrometry:
Reference Materials
Alternative Names:
BN-104; BNM-1192; Menin-MLL inhibitor 27
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Zefamenib (BN-104) is an effective selective brain membrane protein inhibitor with oral activity, and it's also a Menin inhibitor, it can block the Menin-MLL interaction and leads to the degradation of Menin protein. Zefamenib is a weak hERG inhibitor, with an IC50 greater than 100 µM. Zefamenib has anti-tumor activity and can be used in cancer research, such as for acute myeloid leukemia[1].