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T863

Catalogue number:
HY-32219-25mg
Supplier:
Size:
25 mg
Product is available in:
  • UK
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

701232-20-4

Purity:

99.83

Molecular Formula:

C22H26N4O3

Molecular Weight:

394.47

Mass Spectrometry:

Reference Materials

Product Description:

T863 is an orally active, selective and potent DGAT1 (acyl-CoA:diacylglycerol acyltransferase 1) inhibitor with an IC50 of 15 nM. T863 has no inhibitory activity against human MGAT3, human DGAT2, or human MGAT2. T863 interacts with the acyl-CoA binding site of DGAT1, and inhibits triacylglycerol synthesis in cells[1][2].