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CCT241736

Catalogue number:
HY-18161-10mg
Supplier:
Size:
10 mg
Product is available in:
  • UK
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1402709-93-6

Purity:

99.88

Molecular Formula:

C22H23Cl2N7

Molecular Weight:

456.37

Mass Spectrometry:

Reference Materials

Product Description:

CCT241736 is a potent and orally bioavailable dual FLT3 and Aurora kinase inhibitor, which inhibits Aurora kinases (Aurora-A Kd, 7.5 nM, IC50, 38 nM; Aurora-B Kd, 48 nM), FLT3 kinase (Kd, 6.2 nM), and FLT3 mutants including FLT3-ITD (Kd, 38 nM) and FLT3(D835Y) (Kd, 14 nM).