Linaprazan glurate
Catalogue number:
HY-145578-25mg
Supplier:
Size:
25 mg
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1228559-81-6
Purity:
99.67
Molecular Formula:
C26H32N4O5
Molecular Weight:
480.56
Mass Spectrometry:
Reference Materials
Alternative Names:
X842
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Linaprazan glurate (X842) is an orally atcive prodrug of Linaprazan (HY-100412) with a potent and prolonged inhibitory effect on gastric acid secretion. Linaprazan glurate is rapidly transformed by enzymatic cleavage into its active metabolite, linaprazan. Linaprazan glurate is a potassium-competitive acid blocker. Linaprazan glurate selectively inhibites acid formation from gastric H⁺/K⁺-ATPase in a potassium-dependent manner (IC₅₀ = 436.2 nM). Linaprazan glurate can be used for the studies of erosive esophagitis (EE)[1][2].