Opiranserin (hydrochloride)
Catalogue number:
HY-109067A-1mL
Supplier:
Size:
1 ml
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1440796-75-7
Purity:
99.62
Molecular Formula:
C21H35ClN2O5
Molecular Weight:
430.97
Mass Spectrometry:
Reference Materials
Alternative Names:
VVZ-149 (hydrochloride)
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- MSDS: View or download
- Protocol: View or download
Product Description:
Opiranserin (VVZ-149) hydrochloride, a non-opioid and non-NSAID analgesic candidate, is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 µM, respectively. Opiranserin hydrochloride shows antagonistic activity on rP2X3 (IC50=0.87 µM). Opiranserin hydrochloride is development as an injectable agent for the treatment of postoperative pain[1][2][3]. 10mM