Relugolix
Catalogue number:
HY-16474-100mg
Supplier:
Size:
100 mg
Product is available in:
£630.00
Special price until 31 Dec 2025
Normal price £700.00
Shipping is calculated in checkout
Normal price £700.00
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
737789-87-6
Purity:
99.67
Molecular Formula:
C29H27F2N7O5S
Molecular Weight:
623.63
Alternative Names:
TAK-385
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Relugolix (TAK-385) is a potent, orally active, nonpeptidic gonadotropin-releasing hormone (GnRH) antagonist. Relugolix possesses high affinity and potent antagonistic activity for human receptor (binding IC50=0.33 nM) and monkey receptor (IC50=0.32 nM) compared with TAK-013 (HY-100209)[1]. Relugolix is used for the study of sex-hormone-dependent diseases, such as including endometriosis, uterine fibroids and prostate cancer et al[2].