Inobrodib
Catalogue number:
HY-111784-1mL
Supplier:
Size:
1 ml
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
2222941-37-7
Purity:
99.94
Molecular Formula:
C30H32F2N4O3
Molecular Weight:
534.60
Mass Spectrometry:
Reference Materials
Alternative Names:
CCS1477
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
Inobrodib (CCS1477) is an orally active, potent, and selective inhibitor of the p300/CBP bromodomain. Inobrodib binds to p300 and CBP with Kd values of 1.3 and 1.7 nM, respectively, and with 170/130-fold selectivity compared with BRD4 with a Kd of 222 nM. CCS1477 inhibits cell proliferation in prostate cancer cell lines and decreases androgen receptor (AR)- and C-MYC-regulated gene expression[1]. 10mM