Asimadoline (hydrochloride)
Catalogue number:
HY-107384A-25mg
Supplier:
Size:
25 mg
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
185951-07-9
Purity:
99.82
Molecular Formula:
C27H31ClN2O2
Molecular Weight:
451.00
Mass Spectrometry:
Reference Materials
Alternative Names:
EMD-61753 (hydrochloride)
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- MSDS: View or download
- Protocol: View or download
Product Description:
Asimadoline (EMD-61753) hydrochloride is an orally active, selective and peripherally active κ-opioid agonist with IC50s of 5.6 nM (guinea pig) and 1.2 nM (human recombinant). Asimadoline hydrochloride has low permeability across the blood brain barrier and has peripheral anti-inflammatory actions. Asimadoline hydrochloride ameliorates allodynia in diabetic rats and has the potential for irritable bowel syndrome (IBS)[1][2][3].