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Facinicline (hydrochloride)

Catalogue number:
HY-108057A-10mg
Supplier:
Size:
10 mg
Product is available in:
  • UK
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

677305-02-1

Purity:

99.66

Molecular Formula:

C15H19ClN4O

Molecular Weight:

306.79

Mass Spectrometry:

Reference Materials

Alternative Names:

RG3487 (hydrochloride)

Product Description:

Facinicline hydrochloride (RG3487 hydrochloride) is an orally active nicotinic α7 receptor partial agonist, with a Ki of 6 nM for α7 human nAChR. Facinicline hydrochloride (RG3487 hydrochloride) improves cognition and sensorimotor gating in rodents. Facinicline hydrochloride (RG3487 hydrochloride) shows high affinity (antagonist) to 5-HT3Rs with a Ki value of 1.2 nM[1].