SR 144528
Catalogue number:
CAY9000491-10 mg
Supplier:
Size:
10 mg
Product is available in:
£310.00
Estimated delivery Tue 6 Jan
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
192703-06-3
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Formula:
C29H34ClN3O
Molecular Weight:
476.1
Alternative Names:
5-
- MSDS: View or download
Product Description:
A CB2 receptor antagonist (Ki = 0.6 nM); selective for CB2 over CB1 receptors in CHO cells expressing human receptors (Ki = 437 nM); reverses CP 55,940-induced inhibition of forskolin-induced adenylyl cyclase activity in CHO cells expressing human CB2 receptors (EC50 = 10 nM); reduces paw swelling in a mouse model of carrageenin-induced paw edema at 0.01 mg/kg
