Immepip (hydrobromide)
Catalogue number:
CAY29518-10 mg
Supplier:
Size:
10 mg
Product is available in:
£223.00
Estimated delivery Wed 15 Apr
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
164391-47-3
Purity:
≥95%
Formulation:
A crystalline solid
Molecular Formula:
C9H15N3 • 2HBr
Molecular Weight:
327.0595
Alternative Names:
4-(1h-
Product Description:
A histamine H3 receptor agonist (KI = 0.4 nM in SK-N-MC cell membranes expressing the human receptor); selective for histamine H3 over H1 and H2 receptors in CHO cell membranes expressing the guinea pig and human receptors, respectively (Kis = >16 µM for both) but also agonizes H4 receptors (KI = 9 nM in SK-N-MC cell membranes expressing the human receptor); decreases hypothalamic histamine release in anesthetized rats at 5 mg/kg; decreases flinching in the formalin test in rats at 5 and 30 mg/kg and inhibits formalin-induced paw edema at 30 mg/kg
