Cytisine
Catalogue number:
CAY26437-500 mg
Supplier:
Size:
500 mg
Product is available in:
£571.00
Estimated delivery Fri 10 Apr
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
485-35-8
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Formula:
C11H14N2O
Molecular Weight:
190.24174
Alternative Names:
(1r,5s)-
- MSDS: View or download
Product Description:
An alkaloid and a partial agonist of nAChRs (EC50 = 1 µM for α4β2 subunit-containing nAChRs expressed in Xenopus oocytes); inhibits current induced by acetylcholine by 50% in Xenopus oocytes expressing α4β2-subunit containing nAChRs at 20 nM; binds to α2β2, α2β4, α3β2, α3β4, α4β2, and α4β4 nAChR subunits (Kis = 1.1, 5.4, 37, 220, 1.5, and 2.1 nM, respectively); reduces increases in the ICSS threshold of nicotine-withdrawing rats at 3 mg/kg
