FR122047 (hydrochloride)
Catalogue number:
CAY10039-5 mg
Supplier:
Size:
5 mg
Product is available in:
£109.00
Estimated delivery Thu 23 Jul
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
130717-51-0
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Formula:
C23H25N3O3S • HCl
Molecular Weight:
459.98966
Alternative Names:
1-
Product Description:
A selective COX-1 inhibitor (IC50 = 0.028 µM for the human enzyme); selective for COX-1 over COX-2 (IC50 = 65 µM); inhibits arachidonic acid, collagen, and ADP-induced platelet aggregation in human platelet-rich plasma (IC50 = 180-200 nM); unlike aspirin, it does not induce gastric damage at 100 mg/kg, p.o.; has an anti-inflammatory effect in a rat models of collagen-induced arthritis
