LUF6283
Catalogue number:
CAY15423-5 mg
Supplier:
Size:
5 mg
Product is available in:
£131.00
Estimated delivery Wed 15 Apr
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
92933-48-7
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Formula:
C8H12N2O2
Molecular Weight:
168.2
Alternative Names:
5-butyl-1h-
Product Description:
A partial agonist of GPR109A/HCA2 receptors (Ki = 0.55 µM in a radioligand binding assay); stimulates [35S]-GTPγS binding and increases phosphorylation of ERK in HEK293T cells expressing GPR109A/HCA2 receptors (EC50s = 3.1 and 0.32 µM, respectively); reduces plasma levels of VLDL and hepatic expression of apolipoprotein B in mice at 400 mg/kg per day
