GSK180736A
Catalogue number:
CAY26182-5 mg
Supplier:
Size:
5 mg
Product is available in:
£131.00
Estimated delivery Thu 25 Dec
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
817194-38-0
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Formula:
C19H16FN5O2
Molecular Weight:
365.361243
Alternative Names:
4-(4-fluoro
Product Description:
A ROCK1 and GRK2 inhibitor (IC50s = 14 and 0.77 µM, respectively); selective for GRK2 over GRK1, GRK5, and PKA (IC50 = >100 µM for all); selective for ROCK1 over RSK1 and p20S6K (IC50s = 3,100 and 2,850 nM, respectively); increases maximum contractility in isolated mouse cardiomyocytes at 1 µM
