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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1433497-19-8
Purity:
≥95%
Formulation:
A crystalline solid
Molecular Weight:
578.7
Alternative Names:
4-[5-[3,5-bis(1,1-dimethylethyl)phenyl]-1-[4-[(4-methyl-1-piperazinyl)carbonyl]phenyl]-1h-pyrazol-3-yl]-benzoic acid
- Data sheet: View or download
- MSDS: View or download
Product Description:
A potent RARγ antagonist (Ki = 1.1 nM); selective for RARγ over RARα and RARβ (Kis = >1,700 and >2,980 nM, respectively); reduces differential weight bearing between the contralateral and ipsilateral limbs in a rat model of monoiodoacetate-induced osteoarthritis (ED50 = 0.72 mg/kg)
Storage Temperature:
-20°C