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SAfit2

Catalogue number:
CAY24366-5 mg
Supplier:
Size:
5 mg
Product is available in:
  • UK
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£1155.00 Estimated delivery Mon 20 Apr
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1643125-33-0

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Formula:

C46H62N2O10

Molecular Weight:

802.99196

Alternative Names:

(2s)-1-[(2s)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]-2-piperidinecarboxylic acid, (1r)-3-(3,4-dimethoxyphenyl)-1-[3-[2-(4-morpholinyl)ethoxy]phenyl]propyl ester

Product Description:

An FKBP51 inhibitor (Ki = 6 nM); highly selective for FKBP51 over FKBP52 (Ki = >50,000 nM); decreases plasma corticosterone levels to a greater extent than control mice following dexamethasone administration (20 mg/kg); does not increase plasma corticosterone levels as high as in control mice following administration of CRF (20 mg/kg); has antidepressant-like and anxiolytic-like activity in mice (20 mg/kg)

CAY24366-5 mg: SAfit2
CAY24366-5 mg: SAfit2