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Ketanserin (tartrate)

Catalogue number:
CAY22058-100 mg
Supplier:
Size:
100 mg
Product is available in:
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£88.00 Estimated delivery Wed 24 Dec
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

83846-83-7

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Formula:

C22H22FN3O3 • C4H6O6

Molecular Weight:

545.5

Alternative Names:

3-[2-[4-(4-fluorobenzoyl)-1-piperidinyl]ethyl]-2,4(1h,3h)-quinazolinedione (2r,3r)-2,3-dihydroxybutanedioate

Product Description:

A potent 5-HT2 receptor antagonist (IC50 = 6.3 nM; Ki = 2.1 nM); has activity at H1, α1-ARs, and DA receptors; Kis = 10, 10, and 220 nM, respectively); induces dose-dependent inhibition of contractile responses to 5-HT in arteries and veins; significantly decreases BP, BPV, and hypertensive organ damage in spontaneously hypertensive rats

CAY22058-100 mg: Ketanserin (tartrate)
CAY22058-100 mg: Ketanserin (tartrate)