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Vorapaxar

Catalogue number:
CAY23119-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
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£80.00 Estimated delivery Wed 15 Apr
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

618385-01-6

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Formula:

C29H33FN2O4

Molecular Weight:

492.6

Alternative Names:

n-[(1r,3ar,4ar,6r,8ar,9s,9as)-9-[(1e)-2-[5-(3-fluorophenyl)-2-pyridinyl]ethenyl]dodecahydro-1-methyl-3-oxonaphtho[2,3-c]furan-6-yl]-carbamic acid, ethyl ester

Product Description:

A PAR1 antagonist (Ki = 8.1 nM); selective for PAR1 over other PARs, as well as a number of GPCRs, ion channels, and receptors; inhibits thrombin- and haTRAP-induced platelet aggregation (IC50s = 47 and 25 nM, respectively); completely inhibits platelet aggregation in cynomolgus monkeys ex vivo when used at a dose of 0.1 mg/kg i.v.

CAY23119-1 mg: Vorapaxar
CAY23119-1 mg: Vorapaxar