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Raxatrigine (hydrochloride)

Catalogue number:
CAY23490-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
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£52.00 Estimated delivery Tue 14 Apr
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

934240-31-0

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Formula:

C18H19FN2O2 • HCl

Molecular Weight:

350.8

Alternative Names:

(2s)-5r-[4-[(2-fluorophenyl)methoxy]phenyl]-2-pyrrolidinecarboxamide, monohydrochloride, biib074, cnv1014802, gsk1014802a, vixotrigine

Product Description:

An inhibitor of voltage-gated sodium channels (IC50s = 22, 13, 23, 10, 84, 15, 32, and 6 µM for Nav1.1- Nav1.8 channels); has state-dependent activity at the Nav1.7 channel (IC50s = 6.3 and 54 µM for open/inactivated and closed/resting states); decreases pain behavior in an OD1 mouse pain model

CAY23490-1 mg: Raxatrigine (hydrochlorid
CAY23490-1 mg: Raxatrigine (hydrochloride)