Linagliptin
Catalogue number:
CAY23306-500 mg
Supplier:
Size:
500 mg
Product is available in:
£152.00
Estimated delivery Wed 24 Dec
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
668270-12-0
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Formula:
C25H28N8O2
Molecular Weight:
472.5
Alternative Names:
8-[(3r)-3-
Product Description:
A potent DPP-4 inhibitor (IC50 = 1 nM for human recombinant DPP-4); ≥10,000-fold selectivity for DPP-4 over other a panel of 11 peptidases and proteases; inhibits 90% of plasma DPP-4 activity in rat; dose-dependently decreases plasma glucose and increases plasma levels of GLP-1 and insulin in Zucker diabetic fatty rats; reduces HbA1c levels in mice with high-fat diet- and low-dose streptozotocin-induced diabetes
