CPI-637
Catalogue number:
CAY23500-10 mg
Supplier:
Size:
10 mg
Product is available in:
£236.00
Estimated delivery Wed 15 Apr
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1884712-47-3
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Formula:
C22H22N6O
Molecular Weight:
386.5
Alternative Names:
(4r)-1,3,4,5-
Product Description:
An inhibitor of CBP/EP300 bromodomains (IC50s = 30 and 51 nM in a TR-FRET assay); selective for CBP and EP300 over the BET family of bromodomains (IC50s = >10 µM); is active at bromodomain BRD9 (IC50 = 0.73 µM); inhibits CBP (IC50 = 0.3 µM in a BRET assay) and inhibits MYC expression (EC50 = 0.6 µM) in AMO-1 cells
