Cisapride
Catalogue number:
CAY21657-10 mg
Supplier:
Size:
10 mg
Product is available in:
£107.00
Estimated delivery Wed 17 Sep
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
81098-60-4
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Formula:
C23H29ClFN3O4
Molecular Weight:
466
Alternative Names:
rel-4-amino-5-chloro-n-[1-[(3r,4s)-3-(4-fluorophenoxy)propyl]-3-methoxy-4-piperidinyl]-2-methoxy-benzamide
Product Description:
A 5-HT4 receptor agonist (IC50 = 0.483 µM in COS-7 cells expressing the human receptor); induces relaxation of precontracted isolated rat esophageal thoracic muscularis mucosae preparations (EC50 = 102.33 nM); increases the rate of gastric emptying in rats at (0.5 mg/kg); an hERG channel blocker; bind to hERG channels (IC50 = <1 µM in a fluorescence polarization assay)
