Glucagon Receptor Antagonist 4
Catalogue number:
CAY22164-10 mg
Supplier:
Size:
10 mg
Product is available in:
£214.00
Estimated delivery Mon 29 Sep
Shipping is calculated in checkout
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1393124-08-7
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Formula:
C26H28F3N3O4
Molecular Weight:
503.5
Alternative Names:
n-[4-[(1s)-1-[3,5-dimethyl-4-[4-(trifluoromethyl)-1h-pyrazol-1-yl]phenoxy]butyl]benzoyl]-β-alanine, gcgr antagonist iv
- Data sheet: View or download
- MSDS: View or download
Product Description:
A GCGR antagonist (Ki = 14 nM for the human recombinant receptor); greater than 230-fold selective for GCGR over the GLP-1 receptor, as well as a panel of 69 receptors, ion channels, uptake sites, and enzymes at 10 µM; prevents glucagon-induced increases in glucose levels in rat blood at 7.5 and 75 mg/kg
