Glucagon Receptor Antagonist 4
Catalogue number:
CAY22164-10 mg
Supplier:
Size:
10 mg
Product is available in:
£236.00
Estimated delivery Wed 8 Apr
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1393124-08-7
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Formula:
C26H28F3N3O4
Molecular Weight:
503.5
Alternative Names:
n-[4-[(1s)-1-
- MSDS: View or download
Product Description:
A GCGR antagonist (Ki = 14 nM for the human recombinant receptor); greater than 230-fold selective for GCGR over the GLP-1 receptor, as well as a panel of 69 receptors, ion channels, uptake sites, and enzymes at 10 µM; prevents glucagon-induced increases in glucose levels in rat blood at 7.5 and 75 mg/kg
