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MJN110

Catalogue number:
CAY17583-25 mg
Supplier:
Size:
25 mg
Product is available in:
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£509.00 Estimated delivery Tue 19 May
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1438416-21-7

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Formula:

C22H21Cl2N3O4

Molecular Weight:

462.3

Alternative Names:

4-[bis(4-chlorophenyl)methyl]-1-piperazinecarboxylic acid, 2,5-dioxo-1-pyrrolidinyl ester, 2,5-dioxopyrrolidin-1-yl 4-[bis(4-chlorophenyl)methyl]piperazine-1-carboxylate

Product Description:

An inhibitor of MAGL (IC50 = 9.1 nM) and to a lesser extent ABHD6 with potent selectivity over FAAH (IC50 > 10 µM) and other brain serine hydrolases; inhibits 2-AG hydrolysis (IC50 = 2.1 nM) with no effect on AEA hydrolysis up to 50 µM; alleviates mechanical allodynia in a rat model of diabetic neuropathy at 5 mg/kg

CAY17583-25 mg: MJN110
CAY17583-25 mg: MJN110