LEI-106
Catalogue number:
CAY16419-5 mg
Supplier:
Size:
5 mg
Product is available in:
£169.00
Estimated delivery Wed 5 Nov
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1620582-23-1
Alternative Names:
n-[(3,4-dihydro-2,2-dimethyl-2h-1-benzopyran-6-yl)sulfonyl]-n-[(4-phenoxyphenyl)methyl]-glycine
Product Description:
A potent in vitro inhibitor of sn-1 DAGLα (IC50 = 18 nM); blocks the hydrolysis of sn-1-oleoyl-2-AG, the natural substrate of DAGLα, with a Ki value of 0.7 µM; inhibits the hydrolysis of 2-AG by the monoacylglycerol lipase ABHD6 in membrane preparations (Ki = 0.8 µM)
