Cariporide
Catalogue number:
CAY16935-5 mg
Supplier:
Size:
5 mg
Product is available in:
£88.00
Estimated delivery Wed 15 Apr
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
159138-80-4
Purity:
≥95%
Formulation:
A crystalline solid
Molecular Formula:
C12H17N3O3S
Molecular Weight:
283.3
Alternative Names:
n-
Product Description:
An NHE-1 inhibitor (IC50 = 0.56 µM in an intracellular pH recovery assay); selective for NHE-1 over NHE-2 (IC50 = 28 µM in an intracellular pH recovery assay); inhibits sodium propionate-induced swelling of isolated human platelets (IC50 = 0.023 µM); reduces the myocardial infarct size as a percentage of the area at risk in a rabbit model of ischemia-reperfusion injury induced by coronary artery occlusion at 1 mg/kg; decreases ventricular tachycardia duration in a rat model of coronary artery ligation and reperfusion-induced arrhythmia at 1 mg/kg




