Metoprolol (succinate)
Catalogue number:
CAY15429-100 mg
Supplier:
Size:
100 mg
Product is available in:
£582.00
Estimated delivery Tue 9 Jun
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
98418-47-4
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Formula:
C15H25NO3 • 1/2C4H6O4
Molecular Weight:
326.4
Alternative Names:
butanedioic acid, compd. with 1-[4-(2-meth
Product Description:
A β1-AR antagonist (Ki = 47 nM in CHO cells expressing the human receptor); selective for β1- over β2- and β3-ARs (Kis = 2,730 and >10,000 nM, respectively, in CHO cells expressing the human receptors); reduces GTP-induced AC activity in CHO cells expressing β1- and β2-ARs at 4.7 µM; reduces the pulse rate in isolated rat atria in a concentration-dependent manner; reduces increased heart rate and MAP at 30 mg/kg in a rat model of systolic hypertension induced by a fructose-rich diet
