GSK-J1 (sodium salt)
Catalogue number:
CAY12054-5 mg
Supplier:
Size:
5 mg
Product is available in:
£147.00
Estimated delivery Tue 7 Oct
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1797832-71-3
Purity:
≥95%
Formulation:
A crystalline solid
Molecular Formula:
C22H22N5O2 • Na
Molecular Weight:
411.4
Alternative Names:
n-[2-(2-pyridinyl)-6-(1,2,4,5-tetrahydro-3h-3-benzazepin-3-yl)-4-pyrimidinyl]-β-alanine, monosodium salt
Product Description:
A potent, cell impermeable inhibitor of the H3K27 histone demethylases JMJD3 and UTX (IC50s = 18 and 56 µM, respectively as measured by mass spectrometry; IC50 = 60 nM in JMJD3 antibody-based assays)