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GSK-J4 (hydrochloride)

Catalogue number:
CAY12073-5 mg
Supplier:
Size:
5 mg
Product is available in:
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£73.00 Estimated delivery Wed 24 Dec
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1797983-09-5

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Formula:

C24H27N5O2 • HCl

Molecular Weight:

454

Alternative Names:

n-[2-(2-pyridinyl)-6-(1,2,4,5-tetrahydro-3h-3-benzazepin-3-yl)-4-pyrimidinyl]-β-alanine, ethyl ester, monohydrochloride

Product Description:

An ethyl ester prodrug of the JMJD3 selective histone demethylase inhibitor GSK-J1; reduces LPS-induced proinflammatory cytokine production, including that of TNFα (IC50 = 9 µM) in human primary macrophages

CAY12073-5 mg: GSK-J4 (hydrochloride)
CAY12073-5 mg: GSK-J4 (hydrochloride)