GSK1059615
Catalogue number:
CAY11569-5 mg
Supplier:
Size:
5 mg
Product is available in:
£118.00
Estimated delivery Wed 17 Dec
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
958852-01-2
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Formula:
C18H11N3O2S
Molecular Weight:
333.4
Alternative Names:
5z-[[4-(4-
Product Description:
A potent, reversible, ATP-competitive, thiazolidinedione inhibitor of PI3Kα (IC50 = 2 nM) and the common activating mutants of p100α (E542K, E545K, and H1047R) found in cancer; prevents proliferation in BT474 tumor xenografts and reduces MAPK signaling with twice daily dosing at 25 mg/kg
