GSK1059615
Catalogue number:
CAY11569-5 mg
Supplier:
Size:
5 mg
Product is available in:
£131.00
Estimated delivery Fri 8 May
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
958852-01-2
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Formula:
C18H11N3O2S
Molecular Weight:
333.4
Alternative Names:
5z-[[4-(4-
Product Description:
A potent, reversible, ATP-competitive, thiazolidinedione inhibitor of PI3Kα (IC50 = 2 nM) and the common activating mutants of p100α (E542K, E545K, and H1047R) found in cancer; prevents proliferation in BT474 tumor xenografts and reduces MAPK signaling with twice daily dosing at 25 mg/kg
