Tazemetostat trihydrochloride
Catalogue number:
T15240-50 mg
Supplier:
Size:
50 mg
Product is available in:
CAS Number:
1403255-00-4
Molecular Formula:
C34H47Cl3N4O4
Molecular Weight:
682.12
Alternative Names:
EPZ-6438 trihydrochloride , E-7438 trihydrochloride
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Product Description:
Tazemetostat trihydrochloride is a selective and orally available inhibitor of EZH2 (IC50: 4 nM for rat EZH2). It inhibits the activity of human PRC2-containing wild-type EZH2 (Ki: 2.5 nM). It inhibits EZH2 (IC50s: 11 and 16 nM in peptide assay and nucleosome assay).