PSB-06126
Catalogue number:
CAY42173-25 mg
Supplier:
Size:
25 mg
Product is available in:
£441.00
Estimated delivery Fri 9 Jan
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1052089-16-3
Purity:
≥95%
Formulation:
A solid
Molecular Formula:
C24H15N2O5S • Na
Molecular Weight:
466.44215
Alternative Names:
1-amino-9,10-
Product Description:
An inhibitor of NTPDase 3 (IC50 = 1.5 µM for the rat enzyme); selective for NTPDase 3 over NTPDase 1 and -2 at 1 mM; activates KCa/BK channels in rabbit bladder smooth muscle preparations in an inside/out patch-clamp assay (EC50 = 0.841 µM); inhibits UTP-induced calcium mobilization in 1321N1 cells expressing the human purinergic P2Y4 receptor (IC50 = 7.72 µM); selectively increases extracellular ATP levels in BM-MSCs isolated from postmenopausal women over those from young women at 3 µM; increases matrix mineralization in primary postmenopausal women BM-MSCs