PSB-06126
Catalogue number:
CAY42173-25 mg
Supplier:
Size:
25 mg
Product is available in:
£400.00
Estimated delivery Tue 16 Dec
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1052089-16-3
Purity:
≥95%
Formulation:
A solid
Molecular Formula:
C24H15N2O5S • Na
Molecular Weight:
466.44215
Alternative Names:
1-amino-9,10-
Product Description:
An inhibitor of NTPDase 3 (IC50 = 1.5 µM for the rat enzyme); selective for NTPDase 3 over NTPDase 1 and -2 at 1 mM; activates KCa/BK channels in rabbit bladder smooth muscle preparations in an inside/out patch-clamp assay (EC50 = 0.841 µM); inhibits UTP-induced calcium mobilization in 1321N1 cells expressing the human purinergic P2Y4 receptor (IC50 = 7.72 µM); selectively increases extracellular ATP levels in BM-MSCs isolated from postmenopausal women over those from young women at 3 µM; increases matrix mineralization in primary postmenopausal women BM-MSCs