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CVN293

Catalogue number:
CAY40983-10 mg
Supplier:
Size:
10 mg
Product is available in:
  • UK
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£628.00 Estimated delivery Wed 24 Dec
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

2815296-08-1

Purity:

≥98%

Formulation:

A solid

Molecular Formula:

C14H10FN7O

Molecular Weight:

311.274183

Alternative Names:

4-[7-fluoro-1-(3-pyridazinylmethyl)-1h-benzimidazol-2-yl]-1,2,5-oxadiazol-3-amine

Product Description:

A K2P13.1/THIK1 channel inhibitor (IC50 = 49 nM); selective for K2P13.1/THIK1 over K2P6.1/TWIK2 and K2P2.1/TREK-1 channels (IC50s = >30,000 nM for both); inhibits NLRP3 inflammasome-mediated IL-1β production in LPS-stimulated primary neonatal murine microglia (IC50 = 24 nM)