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CJ-42794

Catalogue number:
T14975-25 mg
Size:
25 mg
Product is available in:
  • UK
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CAS Number:

847728-01-2

Purity:

≥98%

Molecular Formula:

C22H17ClFNO4

Molecular Weight:

413.83

Alternative Names:

CJ-042794

Product Description:

CJ-42794 (CJ-042794) is a selective antagonist of the prostaglandin E receptor subtype 4 (EP4), inhibiting [3H]-PGE2 binding to the human EP4 receptor with a mean pKi of 8.5. It exhibits a binding affinity that is at least 200-fold more selective for the human EP4 receptor than for other human EP receptor subtypes (EP1, EP2, and EP3) (IC50: 8.5 (pKi)).