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GSK180736A

Catalogue number:
T3513-1 mL
Size:
1 ml * 10 mM (in dmso)
Product is available in:
  • UK
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CAS Number:

817194-38-0

Purity:

≥98%

Molecular Formula:

C19H16FN5O2

Molecular Weight:

365.36

Alternative Names:

GSK180736

Product Description:

GSK180736A is an effective and selective GRK2 inhibitor (IC50: 0.77 µM) and >100-fold selectivity over other GRKs. It is a weak inhibitor of PKA (IC50: 30 µM), but highly effective against ROCK1 (IC50: 100 nM).