PBRM1-BD2-IN-2
Catalogue number:
T60156-10 mg
Supplier:
Size:
10 mg
Product is available in:
CAS Number:
2819989-57-4
Purity:
≥98%
Molecular Formula:
C14H9Cl2FN2O
Molecular Weight:
311.14
- Data sheet: View or download
- MSDS: View or download
- Protocol: View or download
Product Description:
PBRM1-BD2-IN-2, a selective and cell-active inhibitor of the polybromo-1 (PBRM1) bromodomain, exhibits binding affinity and inhibitory activity specifically targeting the PBRM1-BD2 domain, with Kd and IC50 values of 9.3 µM and 1.0 µM, respectively. This compound is utilized in cancer research.