PF 429242
Catalogue number:
T4317-1 mg
Supplier:
Size:
1 mg
Product is available in:
CAS Number:
947303-87-9
Purity:
≥98%
Molecular Formula:
C25H35N3O2
Molecular Weight:
409.56
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- MSDS: View or download
Product Description:
PF-429242 is a competitive inhibitor of sterol regulatory element-binding protein (SREBP) site 1 protease (IC50 = 0.175 µM). It is selective for site 1 protease against a panel of serine proteases. PF-429242 inhibits rate of cholesterol synthesis in CHO cells (IC50 = 0.53 µM).