GNE-207
Catalogue number:
T15399-100 mg
Supplier:
Size:
100 mg
Product is available in:
CAS Number:
2158266-58-9
Molecular Formula:
C29H30N6O3
Molecular Weight:
510.59
- Data sheet: View or download
- MSDS: View or download
Product Description:
GNE-207 is a selective and orally bioavailable inhibitor of the bromodomain of CBP (IC50: 1 nM). It has a selective index of >2500-fold against BRD4 (1). GNE-207 displays excellent CBP potency (EC50: 18 nM for MYC expression in MV-4-11 cells).
