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AZD 5462

Catalogue number:
CAY40956-500 ug
Supplier:
Size:
500 µg
Product is available in:
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£185.00 Estimated delivery Wed 15 Apr
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

2787501-83-9

Purity:

≥98%

Formulation:

A solid

Molecular Formula:

C30H41FN2O6

Molecular Weight:

544.7

Alternative Names:

cis-4-[2-fluoro-4-methoxy-5-[[[(1s,2r,3s,4r)-3-[[[(1-methylcyclobutyl)methyl]amino]carbonyl]bicyclo[2.2.1]hept-2-yl]amino]carbonyl]phenoxy]-1-methyl-cyclohexane

Product Description:

An RXFP1 agonist; induces cAMP mobilization in HEK293 cells expressing the human RXFP1 (EC50 = 15.85 nM); increases heart rate and MABP in rats; increases the left ventricular ejection fraction (LVEF) in a cynomolgus monkey model of heart failure induced by a high-fat diet and age at 1 or 10 mg/kg per day