MYCi975
Catalogue number:
CAY39622-5 mg
Supplier:
Size:
5 mg
Product is available in:
£245.00
Estimated delivery Wed 15 Apr
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
2289691-01-4
Purity:
≥98%
Formulation:
A solid
Molecular Formula:
C25H16Cl2F6N2O2
Molecular Weight:
561.3
Alternative Names:
4′-chloro-6-[(4-
Product Description:
An inhibitor of the Myc-MAX protein-protein interaction; binds to Myc (Kd = 2.75 µM) and increases GSK3β-mediated Myc phosphorylation in a cell-free assay; decreases the viability of MyC-CaP and LNCaP cells at 5 and 10 µM; induces apoptosis in a panel of 11 breast cancer cell lines at 10 µM; reduces tumor volume in a MyC-CaP mouse xenograft model at 100 mg/kg