KAT8 Inhibitor 19

Name: KAT8 Inhibitor 19
Brand: Cayman Chemical
SKU: CBSKU_201378087
Price: 393 GBP
Availability: InStock

Catalogue number:

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CAY38977-25 mg

Supplier:

Cayman Chemical

Size:

25 mg

Product is available in:

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£393.00

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Estimated delivery Tue 14 Apr
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This product is for research use only and is not for human consumption or therapeutic use.

CAS Number:

28532-21-0

Purity:

≥98%

Formulation:

A solid

Molecular Formula:

C16H13N3O3

Molecular Weight:

295.3

Alternative Names:

4-[4,5-dihydro-3-methyl-5-oxo-4-(1h-pyrrol-2-ylmethylene)-1h-pyrazol-1-yl]-benzoic acid, lysine acetyltransferase 8 inhibitor 19

Product Description:

A KAT8 inhibitor; selective for KAT8 over KAT2A, KAT2B, KAT3B, KAT6A, and KAT7 at 200 µM; reduces H4K16Ac in HT-29 cells at 50 µM; reduces the viability of HCT116, H1299, A549, and U937 cancer cells (IC50s = 39.4, 52.1, 41, and 30.1 µM, respectively)