A2764 (hydrochloride)
Catalogue number:
CAY36943-100 mg
Supplier:
Size:
100 mg
Product is available in:
£288.00
Estimated delivery Wed 15 Apr
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
861038-72-4
Purity:
≥98%
Formulation:
A solid
Molecular Formula:
C15H19ClN2O • 2HCl
Molecular Weight:
351.69822
Alternative Names:
2-[(5-chloro-
Product Description:
An inhibitor of K2P18.1/TRESK (IC50 = 11.8 µM in ionomycin-stimulated Xenopus oocytes expressing the mouse receptor); selective for K2P18.1/TRESK over K2P2.1/TREK1, K2P10.1/TREK2, K2P4.1/TRAAK, K2P3.1/TASK1, K2P3.2/TASK2, K2P3.3/TASK3, K2P16.1/TALK1, and K2P13.1/THIK1 at 100 µM; inhibits basal potassium currents in isolated mouse dorsal root ganglion neurons at 100 µM