Trimeprazine (tartrate)
Catalogue number:
CAY33891-500 mg
Supplier:
Size:
500 mg
Product is available in:
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
4330-99-8
Purity:
≥98%
Formulation:
A solid
Molecular Formula:
C18H22N2S • 1/2C4H6O6
Molecular Weight:
373.5
Alternative Names:
n,n,β-tri
Product Description:
A histamine H1 receptor antagonist (Ki = 0.72 nM in a radioligand binding assay); selective for the histamine H1 receptor over mAChRs (Ki = 38 nM in a radioligand binding assay); inhibits anti-IgE-induced histamine release from isolated human lung fragments (IC50 = 19 nM) but induces histamine release (RC50 = 1.03 µM); reduces SARS-CoV-2 replication in SARS-CoV-2-infected Vero E6 cells (EC50 = 1.76 µM) with a CC50 value of 19.73 µM