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Lumateperone (tosylate)

Catalogue number:
CAY34541-25 mg
Supplier:
Size:
25 mg
Product is available in:
  • UK
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£279.00 Estimated delivery Wed 24 Dec
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1187020-80-9

Purity:

≥95%

Formulation:

A solid

Molecular Formula:

C24H28FN3O • C7H8O3S

Molecular Weight:

565.699763

Alternative Names:

1-(4-fluorophenyl)-4-((6br,10as)-3-methyl-2,3,6b,9,10,10a-hexahydro-1h-pyrido[3',4':4,5]pyrrolo[1,2,3-de]quinoxalin-8(7h)-yl)butan-1-one 4-methylbenzenesulfonic acid, iti-007

Product Description:

An atypical antipsychotic; selectively binds to the 5-HT receptor subtype 5-HT2A over 5-HT1A and 5-HT2C receptors (Kis = 0.54, 1,480, and 173 nM, respectively); binds to dopamine D1, D2, and D4 receptors (Kis = 52, 32, and 108 nM, respectively), α1A- and α1B-adrenergic receptors (Kis = 73 and 31 nM, respectively), and SERT (Ki = 61 nM); reduces quipazine-induced head-twitch behavior in rats (ED50 = 0.12 mg/kg)